ATX inhibitor 1
CAS No. 2225892-70-4
ATX inhibitor 1 ( —— )
产品货号. M22925 CAS No. 2225892-70-4
ATX inhibitor 1 is a potent ATX inhibitor (IC50: 1.23 nM, FS-3 and 2.18 nM, bis-pNPP).
纯度: >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥956 | 有现货 |
|
5MG | ¥1596 | 有现货 |
|
10MG | ¥2527 | 有现货 |
|
25MG | ¥4261 | 有现货 |
|
50MG | ¥6148 | 有现货 |
|
100MG | ¥8667 | 有现货 |
|
200MG | 获取报价 | 有现货 |
|
500MG | 获取报价 | 有现货 |
|
1G | 获取报价 | 有现货 |
|
生物学信息
-
产品名称ATX inhibitor 1
-
注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
-
产品简述ATX inhibitor 1 is a potent ATX inhibitor (IC50: 1.23 nM, FS-3 and 2.18 nM, bis-pNPP).
-
产品描述ATX inhibitor 1 is a potent ATX inhibitor (IC50: 1.23 nM, FS-3 and 2.18 nM, bis-pNPP).
-
同义词——
-
通路Angiogenesis
-
靶点PDE
-
受体ATX
-
研究领域——
-
适应症——
化学信息
-
CAS Number2225892-70-4
-
分子量501.3
-
分子式C21H23Cl2N2O6P
-
纯度>98% (HPLC)
-
溶解度DMSO:250 mg/mL (498.70 mM; Need ultrasonic)
-
SMILESO=P(O)(O)CC1=CC=C(NC(C2CCN(C(OCC3=CC(Cl)=CC(Cl)=C3)=O)CC2)=O)C=C1
-
化学全称——
运输与储存
-
储存条件(-20℃)
-
运输条件With Ice Pack
-
稳定性≥ 2 years
参考文献
1. Balupuri A, et al. Discovery and optimization of ATX inhibitors via modeling, synthesis and biological evaluation. Eur J Med Chem. 2018 Mar 25;148:397-409.
产品手册
关联产品
-
Roflumilast
Roflumilast is a phosphodiesterase-4 (PDE-4) inhibitor.
-
Ginkgolide J
Ginkgolide J has neuroprotective activity it can prevent A beta(1-42) induced inhibition of long-term potentiation in the CA1 region of mouse hippocampal slices.
-
MR-L2
MR-L2 is a reversible and noncompetitive allosteric activator of long-isoform phosphodiesterase-4 (PDE4).